Day 1 – Discovery Chemistry: Latest Case Studies
• Hit to lead optimisation
• Structure-activity relationships
• Optimising allosteric kinase inhibitors
• Fragment based drug discovery
• Combinatorial and high-throughput chemistry
Day 2 – Drug Design: Novel Approaches
• Structure based drug design
• Anti-target modelling
• Protein-ligand interactions
• Antibodies as discovery tools
• Innovation in IPS cell research
• Advances in polypharmacology
• In silico profiling