Invited Speakers: Dr. Petr Kocis, Zeneca Pharmaceuticals
Dr. Shu-Kun Lin, Molecular Diversity Preservation International (MDPI)
Dr. Alisdair MacDonald, Argonaut Technologies, Inc.
Dr. Pierfausto Seneci, GlaxoWellcome S.p.A.
Dr. Jochen Antel, Solvay Pharma
Dr. Anthony Baxter, Oxford Asymmetry International
Prof. Mark Bradley, University of Southampton
Dr. Ernst Bürgisser, Discovery Technologies Ltd.
Dr. Alain Calvet, Parke-Davis Pharmaceutical Research
Dr. Patrick Coffey, Biotage Division of Dyax Corp.
Dr. Ferenc Darvas, ComGenex, Inc.
Dr. Sheila H. DeWitt, Orchid Biocomputer, Inc.
Dr. Simon Fogarty, Cambridge Drug Discovery Ltd.
Dr. Jonathan Frost, Synthelabo Recherche
Dr. Steve Gallion, ArQule, Inc.
Dr. C. John Harris, BioFocus plc
Dr. Peter Hecht, Tripos GmbH
Dr. Karsten Henco, EVOTEC BioSystems
Dr. Nick Jones, Cambridge Combinatorial Chemistry
Dr. John L. Krstenansky, EnzyMed, Inc.
Dr. Hugo Kubinyi, BASF AG
Dr. Aubrey J. Mendonca, IRORI
Dr. Andrea Missio, GlaxoWellcome Medicines Research Centre
Dr. Daniel Obrecht, POLYPHOR Ltd.
Dr. Dieter Poppinger, Novartis Crop Protection AG
Dr. Janice Ramieri, Biotage Division of Dyax Corp.
Program:
Session: Molecular Diversity and Library Design
Novel Combinatorial Chemistry for Drug Lead Discovery
Focused Libraries for Lead Expansion and Optimization: A Toolbox Approach
Molecular Diversity Preservation and Exploitation for Bioactivity Screenings
An Integrated Biocatalytic/Chemical Approach for Bioactive Compounds
Strategies and Technologies for Lead Optimization
In Vivo Leads from Diverse Libraries: New Diversity Approaches
Session: Combinatorial Synthesis
Versatile Resin-Bound Synthons and Traceless Linkers
Synthesis on a Chip
Lead Discovery Using Solid-Phase Chemistry
New Resins and Linkers for Combinatorial Synthesis
Advances in Parallel Synthesis
Chips, Cubes, and Tubes: Taking Library Generation to the Next Level
Solid Supported Synthesis of Protein Epitope-Derived Compound Libraries
An Open, Multivendor Specification for High-Throughput Organic Chemistry (HTOC):
Session: High-Throughput Screening
New FCS-Based Read-Out Technologies for Miniaturized, High-Throughput Applications
Novel Lead Generation through Integrated Target Discovery and HTS
Integrated Discovery with a Novel Automation Concept for HTS
Informatics for HSS and HTS at Novartis Crop Protection
Session: Computational Methodologies and Chemoinformatics
Practical Aspects of the Design and Synthesis of Combinatorial Libraries
Drug Discovery through Synergy: The Full Integration of Chemistry and Informatics
Integration of Combinatorial Chemistry and Structure-Based Drug Design
Similarity and Dissimilarity: A Medicinal Chemist’s View
Design, Analysis, and Comparison of Combinatorial Libraries
Registration :
Please call (617)-630-1352 or email chi@healthtech.com or fax (617)-630-1325
Deadline for Abstracts: 9/18/98
Email for Requests and Registration: chi@healthtech.com